2.3.1.B43: protein-lysine desuccinylase (NAD+)
This is an abbreviated version!
For detailed information about protein-lysine desuccinylase (NAD+), go to the full flat file.
Word Map on EC 2.3.1.B43
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2.3.1.B43
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sirtuins
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sirt3
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deacetylation
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deacetylases
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desuccinylation
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malonylation
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nad-dependent
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sirt1-7
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glutarylation
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diagnostics
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medicine
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drug development
- 2.3.1.B43
- sirtuins
- sirt3
-
deacetylation
- deacetylases
-
desuccinylation
-
malonylation
-
nad-dependent
-
sirt1-7
-
glutarylation
- diagnostics
- medicine
- drug development
Reaction
Synonyms
CobB, CobB Sir2 protein, histone desuccinylase, hSIRT5, hSIRT6, lysine desuccinylase, mitochondrial NAD+-dependent lysine deacylase, NAD+ dependent deacetylase, NAD+-dependent protein deacetylase, NAD+-dependent protein deacylase, NAD+-dependent sirtuin deacetylase, nicotinamide adenine dinucleotide-dependent protein deacetylase, Sir2Af1, SIRT5, SIRT5iso1, SIRT5iso2, SIRT5iso3, SIRT5iso4, sirtuin 5, sirtuin 5 deacylase, sirtuin 5 lysine deacylase, sirtuin deacylase, sirtuin-5, zSIRT5
ECTree
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KM Value
KM Value on EC 2.3.1.B43 - protein-lysine desuccinylase (NAD+)
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0.08018
[histone H2A]-N6-succinyl-L-lysine95
pH 7.5, 37°C, recombinant enzyme
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0.10228
[histone H2A]-N6-succinyl-L-lysine9_(4-15)-A10G peptide
pH 7.5, 37°C, recombinant enzyme
-
0.06173
[histone H2B]-N6-succinyl-L-lysine116
pH 7.5, 37°C, recombinant enzyme
-
0.08777
[histone H2B]-N6-succinyl-L-lysine120
pH 7.5, 37°C, recombinant enzyme
-
0.09973
[histone H2B]-N6-succinyl-L-lysine34
pH 7.5, 37°C, recombinant enzyme
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0.086
[histone H3 K9 peptide]-N6-succinyl-L-lysine
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pH 8.0, 37°C, wild-type enzyme
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0.06051
[histone H3]-N6-succinyl-L-lysine122
pH 7.5, 37°C, recombinant enzyme
-
0.09551
[histone H3]-N6-succinyl-L-lysine14
pH 7.5, 37°C, recombinant enzyme
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0.10442
[histone H3]-N6-succinyl-L-lysine14_(9-20)-A15G peptide
pH 7.5, 37°C, recombinant enzyme
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0.17932
[histone H3]-N6-succinyl-L-lysine56
pH 7.5, 37°C, recombinant enzyme
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0.08489
[histone H3]-N6-succinyl-L-lysine79
pH 7.5, 37°C, recombinant enzyme
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0.07717
[histone H3]-N6-succinyl-L-lysine9
pH 7.5, 37°C, recombinant enzyme
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0.10072
[histone H4]-N6-succinyl-L-lysine12
pH 7.5, 37°C, recombinant enzyme
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0.13153
[histone H4]-N6-succinyl-L-lysine31
pH 7.5, 37°C, recombinant enzyme
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0.06583
[histone H4]-N6-succinyl-L-lysine31_(26-37)-P32A peptide
pH 7.5, 37°C, recombinant enzyme
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0.08268
[histone H4]-N6-succinyl-L-lysine77
pH 7.5, 37°C, recombinant enzyme
-
0.10178
[histone H4]-N6-succinyl-L-lysine91
pH 7.5, 37°C, recombinant enzyme
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0.72
[protein]-N6-acetyl-L-lysine
mutant enzyme Y102A, at 8.0 pH and 25°C
0.069
wild type enzyme, with [protein]-N6-succinyl-L-lysine as cosubstrate, at 8.0 pH and 25°C
0.15
NAD+
cosubstrate: Ac-(N6-succinyl)Lys-7-amido-4-methylcoumarin, pH 8.0, 37°C
0.321
NAD+
mutant enzyme Y102A, with [protein]-N6-succinyl-L-lysine as cosubstrate, at 8.0 pH and 25°C
0.609
NAD+
mutant enzyme R105I, with [protein]-N6-acetyl-L-lysine as cosubstrate, at 8.0 pH and 25°C
1.194
NAD+
mutant enzyme Y102A/R105I, with [protein]-N6-acetyl-L-lysine as cosubstrate, at 8.0 pH and 25°C
1.605
NAD+
mutant enzyme Y102A, with [protein]-N6-acetyl-L-lysine as cosubstrate, at 8.0 pH and 25°C
0.0147
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pH 8.0, 37°C, mutant enzyme Y92F
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0.0151
[histone H3 K9 peptide]-N6-acetyl-L-lysine
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pH 8.0, 37°C, wild-type enzyme
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0.02
[histone H3 K9 peptide]-N6-acetyl-L-lysine
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pH 8.0, 37°C, mutant enzyme R95M
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0.388
[protein]-N6-succinyl-L-lysine
mutant enzyme Y102A/R105I, at 8.0 pH and 25°C
1.658
[protein]-N6-succinyl-L-lysine
mutant enzyme R105I, at 8.0 pH and 25°C