EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.22.B80 | 0.0006 |
- |
(R)-5-amino-2-methyl-N-[1-(naphth-1-yl)ethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.0012 |
- |
(R)-4-amino-2-methyl-N-[1-(naphth-1-yl)ethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.0016 |
- |
(R)-tert-butyl(3-methyl-4-((1-(naphth-1-yl)ethyl)carbamoyl)phenyl)carbamate |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.0023 |
- |
2-methyl-N-[(1R)-naphth-1-ylethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.004 |
- |
(R)-5-(dimethylamino)-2-methyl-N-[1-(naphth-1-yl)ethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.004 |
- |
2-methyl-5-(methylsulfamoyl)-N-[(1R)-1-naphth-1-ylethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.004 |
- |
Disulfiram |
pH 6.5, 30°C, wild-type enzyme, determined in accordance with competitive inhibition |
755817 |
| 3.4.22.B80 | 0.0046 |
- |
(R)-tert-butyl(4-methyl-3-((1-(naphth-1-yl)ethyl)carbamoyl)phenyl)carbamate |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.0048 |
- |
2-methyl-4-[(methylsulfonyl)amino]-N-[(1R)-1-naphth-1-ylethyl]benzamide |
pH 7.5, 25°C |
762930 |
| 3.4.22.B80 | 0.0056 |
- |
7H-furo[3,2-g][1]benzopyran-7-one |
DeISGylation activity, pH 6.8, 37°C |
757319 |
