EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.22.B80 | 0.00015 |
- |
(R)-N-(3-fluorobenzyl)-1-(1-(naphthalen-1-yl)ethyl)-piperidine-4-carboxamide |
pH 7.5, 25°C |
765217 |
| 3.4.22.B80 | 0.00032 |
- |
1-[(R)-1-(1-naphthyl)ethyl]-4-[3,4-(methylenedioxy)benzylamino]carbonylpiperidine |
pH 7.5, temperature not specified in the publication |
765216 |
| 3.4.22.B80 | 0.00034 |
- |
1-[(R)-1-(1-naphthyl)ethyl]-4-(3-methoxybenzylamino)carbonylpiperidine |
pH 7.5, temperature not specified in the publication |
765216 |
| 3.4.22.B80 | 0.00034 |
- |
1-[(R)-1-(1-naphthyl)ethyl]-4-(4-methoxybenzylamino)carbonylpiperidine |
pH 7.5, temperature not specified in the publication |
765216 |
| 3.4.22.B80 | 0.00035 |
- |
(R)-N-((2-methoxypyridin-4-yl)methyl)-1-(1-(naphthalen-1-yl)ethyl)piperidine-4-carboxamide |
pH 7.5, 25°C |
765217 |
| 3.4.22.B80 | 0.00039 |
- |
(R)-N-(3-acetamidobenzyl)-1-(1-(naphthalen-1-yl)ethyl)-piperidine-4-carboxamide |
pH 7.5, 25°C |
765217 |
| 3.4.22.B80 | 0.00044 |
- |
N-[3-fluoro-5-[(1E)-3-[1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidin-4-y]]-3-oxoprop-1-en-1-yl]phenyl}-4-methylpiperazine-1-carboxamide |
20 mM Tris-HCl, 100 mM NaCl, 5 mM 2-hydroxy-1-ethanethiol, pH 7.8, 22°C, synthetic substrate 7-hydroxy-4-methylcoumarin-3-acetyl-RLRGG-NH(CH2)4NH-DABCYL |
762888 |
| 3.4.22.B80 | 0.00046 |
- |
5-(aminomethyl)-2-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide |
pH 7.5, temperature not specified in the publication |
765215 |
| 3.4.22.B80 | 0.00047 |
- |
(R)-N-(4-ethylbenzyl)-1-(1-(naphthalen-1-yl)ethyl)-piperidine-4-carboxamide |
pH 7.5, 25°C |
765217 |
| 3.4.22.B80 | 0.00049 |
- |
(R)-N-(4-fluorobenzyl)-1-(1-(naphthalen-1-yl)ethyl)-piperidine-4-carboxamide |
pH 7.5, 25°C |
765217 |
