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EC Number IC50 Value IC50 Value Maximum Inhibitor Commentary Reference
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - (3-[[2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]methoxy]phenyl)acetic acid KI value is above 5 microM, inhibition profiles are determined by a fluorometric assay with recombinant CAT L employing Z-Phe-Arg-7-amido-4-methylcoumarin as synthetic substrate 696630
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-4-[(6,8-dioxaspiro[3.5]non-7-ylmethyl)amino]-N-methyl-6-[(1-methylpiperidin-4-yl)methoxy]pyrimidine-5-carboxamide IC50 is above 0.001 mM, determined by a fluorometric assay with recombinant catL employing Z-Phe-Arg-7-amido-4-methylcoumarin as synthetic substrate 696641
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-4-[(cyclohexylmethyl)amino]-N-(2-phenylethyl)pyrimidine-5-carboxamide IC50 is above 0.002 mM, inhibition are determined by a fluorometric assay with recombinant Cat L 696638
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-4-[[(4,4-difluorocyclohexyl)methyl]amino]-N-(2-phenylethyl)pyrimidine-5-carboxamide IC50 is above 0.003 mM, inhibition are determined by a fluorometric assay with recombinant Cat L 696638
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-4-[[(4,4-dimethylcyclohexyl)methyl]amino]-N-(2-phenylethyl)pyrimidine-5-carboxamide IC50 is above 0.003 mM inhibition are determined by a fluorometric assay with recombinant Cat L 696638
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-N-(2-phenylethyl)-4-[(spiro[2.5]oct-6-ylmethyl)amino]pyrimidine-5-carboxamide IC50 is above 0.003 mM inhibition are determined by a fluorometric assay with recombinant Cat L 696638
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 2-cyano-N-(4,5-dimethoxybiphenyl-2-yl)-4-[(spiro[2.5]oct-6-ylmethyl)amino]pyrimidine-5-carboxamide IC50 is above 0.003 mM inhibition are determined by a fluorometric assay with recombinant Cat L 696638
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 3-[[2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]methoxy]benzamide KI value is above 1 microM, inhibition profiles are determined by a fluorometric assay with recombinant CAT L employing Z-Phe-Arg-7-amido-4-methylcoumarin as synthetic substrate 696630
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 4-[[2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]methoxy]benzamide KI value is above 1 microM, inhibition profiles are determined by a fluorometric assay with recombinant CAT L employing Z-Phe-Arg-7-amido-4-methylcoumarin as synthetic substrate 696630
Display the word mapDisplay the reaction diagram Show all sequences 3.4.22.15-999 - 4-[[2-cyano-7-(2-cyclohexylethyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]methoxy]benzoic acid KI value is above 2 microM, inhibition profiles are determined by a fluorometric assay with recombinant CAT L employing Z-Phe-Arg-7-amido-4-methylcoumarin as synthetic substrate 696630
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