EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.4.2.12 | 0.0000006 |
- |
N''-cyano-N-[[4-(3,5-difluorobenzene-1-sulfonyl)phenyl]methyl]-N'-pyridin-4-ylguanidine |
pH and temperature not specified in the publication |
735760 |
2.4.2.12 | 0.0000009 |
- |
FK-866 |
i.e. (2E)-N-[4-(1-benzoylpiperidin-4-yl)butyl]-3-phenylprop-2-enamide, pH 7.5, 37°C |
721273 |
2.4.2.12 | 0.0000009 |
- |
N-[4-(4-benzylpiperazine-1-sulfonyl)phenyl]-N'-[(pyridin-3-yl)methyl]thiourea |
at pH 7.5 and 37°C |
737247 |
2.4.2.12 | 0.000001 |
- |
trans-N-(4-((1-Isopropyl-1H-pyrazol-4-yl)sulfonyl)phenyl)-2-(pyridin-3-yl)cyclopropanecarboxamide |
pH and temperature not specified in the publication |
736612 |
2.4.2.12 | 0.0000011 |
- |
trans-N-(4-((1-isopropyl-5-methyl-1H-pyrazol-4-yl)sulfonyl)-phenyl)-2-(pyridin-3-yl)cyclopropanecarboxamide |
pH and temperature not specified in the publication |
736612 |
2.4.2.12 | 0.0000017 |
- |
N''-cyano-N-([4-[6-(morpholin-4-yl)pyridine-3-sulfonyl]phenyl]methyl)-N'-pyridin-4-ylguanidine |
pH and temperature not specified in the publication |
735760 |
2.4.2.12 | 0.0000019 |
- |
N''-cyano-N-[[4-(3-methoxybenzene-1-sulfonyl)phenyl]methyl]-N'-pyridin-4-ylguanidine |
pH and temperature not specified in the publication |
735760 |
2.4.2.12 | 0.000002 |
- |
N''-cyano-N-[[4-(pyridine-3-sulfonyl)phenyl]methyl]-N'-pyridin-4-ylguanidine |
pH and temperature not specified in the publication |
735760 |
2.4.2.12 | 0.000002 |
- |
trans-N-(4-((1-(2-Hydroxy-2-methylpropyl)-1H-pyrazol-4-yl)-sulfonyl)phenyl)-2-(pyridin-3-yl)cyclopropanecarboxamide |
pH and temperature not specified in the publication |
736612 |
2.4.2.12 | 0.0000022 |
- |
N-[[4-(benzenesulfonyl)phenyl]methyl]-N''-cyano-N'-pyridin-3-ylguanidine |
pH and temperature not specified in the publication |
735760 |