EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.13.12.3 | 0.69 |
- |
Indole-3-acetamide |
pH 8.3, 25°C, mutant Y413A |
654683 |
1.13.12.3 | 0.69 |
- |
Indole-3-pyruvate |
pH 8.3, 25°C, mutant Y413A |
654683 |
1.13.12.3 | 4 |
- |
Indole-3-acetamide |
pH 8.3, 25°C, mutant Y413F |
654683 |
1.13.12.3 | 4 |
- |
Indole-3-pyruvate |
pH 8.3, 25°C, mutant Y413F |
654683 |
1.13.12.3 | 13.2 |
- |
Indole-3-acetamide |
pH 8.3, 25°C, wild-type |
654683 |
1.13.12.3 | 13.2 |
- |
Indole-3-pyruvate |
pH 8.3, 25°C, wild-type |
654683 |
1.13.12.3 | 16 |
- |
3-Indoleacetamide |
pH 8.3, 25°C, wild-type |
654682 |
1.13.12.3 | 20 |
- |
3-Indoleacetamide |
pH 8.3, 25°C, mutant R98K |
654682 |
1.13.12.3 | 40 |
- |
3-indolepyruvate |
pH 8.3, 25°C, wild-type |
654682 |
1.13.12.3 | 45 |
- |
3-Indoleacetamide |
pH 8.3, 25°C, mutant R98A |
654682 |