EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.28 | -999 |
- |
more |
inhibition kinetics |
739841 |
1.1.1.28 | 0.12 |
- |
oxalate |
pH 8.0, 30°C |
655064 |
1.1.1.28 | 1.8 |
- |
pyruvate |
pH 7.0, 30°C, recombinant enzyme |
739841 |
1.1.1.28 | 2.8 |
- |
oxamate |
30°C, pH 5.5, wild-type enzyme |
669327 |
1.1.1.28 | 5 |
- |
oxaloacetate |
pH 7.0, 30°C, recombinant enzyme |
739841 |
1.1.1.28 | 19 |
- |
Hydroxypyruvate |
pH 7.0, 30°C, recombinant enzyme |
739841 |
1.1.1.28 | 20 |
- |
pyruvate |
pH 8.0, 30°C, recombinant enzyme, with Mg2+ |
739841 |
1.1.1.28 | 23 |
- |
phenylpyruvate |
pH 7.0, 30°C, recombinant enzyme |
739841 |
1.1.1.28 | 43 |
- |
oxamate |
30°C, pH 5.5, mutant enzyme N97D |
669327 |
1.1.1.28 | 44 |
- |
formate |
30°C, pH 5.5, wild-type enzyme |
669327 |