EC Number |
Inhibitors |
Structure |
---|
3.4.22.B50 | (4E)-1,7-bis(3,4-dihydroxyphenyl)hept-4-en-3-one |
a natural diarylheptanoide inhibitor |
|
3.4.22.B50 | (7R)-5,7-dihydroxy-8-(4-hydroxy-3-methoxyphenyl)-2-(4-hydroxy-4-methylpentyl)-2-methyl-3,4,7,8-tetrahydro-2H,6H-pyrano[3,2-g]chromen-6-one |
a natural geranylated flavonoid inhibitor |
|
3.4.22.B50 | 1,6,6-trimethyl-1,2,6,7,8,9-hexahydrophenanthro[1,2-b]furan-10,11-dione |
a natural tanshinone inhibitor |
|
3.4.22.B50 | 2-methyl-N-[(1R)-1-(naphthalen-2-yl)ethyl]benzamide |
over 90% inhibition at 0.1 mM |
|
3.4.22.B50 | 2-methyl-N-[(1S)-1-(naphthalen-2-yl)ethyl]benzamide |
14% inhibition at 0.1 mM |
|
3.4.22.B50 | 2-methyl-N-[1-(naphthalen-2-yl)ethyl]benzamide |
racemat |
|
3.4.22.B50 | 5-amino-2-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide |
R-isomer, a potent, noncovalent, competitive inhibitor |
|
3.4.22.B50 | 6-Mercaptopurine |
competitive and reversible inhibitor |
|
3.4.22.B50 | 6-Mercaptopurine |
- |
|
3.4.22.B50 | 6-thioguanine |
competitive and reversible inhibitor |
|