EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.1 | -999 |
- |
more |
- |
655804, 656058 |
1.1.1.1 | -999 |
- |
more |
inhibition kinetics |
655206 |
1.1.1.1 | 0.00008 |
- |
caffeic acid |
at 37°C in 0.1 M Na-K phosphate buffer (pH 7.4) |
699982 |
1.1.1.1 | 0.0032 |
- |
4-iodopyrazole |
apparent value |
681763 |
1.1.1.1 | 0.0047 |
- |
4-androsten-3,17-dione |
pH 7.3, 37°C, versus cyclohexanone |
655206 |
1.1.1.1 | 0.0047 |
- |
5alpha-androstan-17beta-ol-3-one |
pH 7.3, 37°C, versus cyclohexanone |
655206 |
1.1.1.1 | 0.0051 |
- |
pyrazole |
at 37°C in 0.1 M Na-K phosphate buffer (pH 7.4) |
699982 |
1.1.1.1 | 0.0079 |
- |
Vanillin |
at 37°C in 0.1 M Na-K phosphate buffer (pH 7.4) |
699982 |
1.1.1.1 | 0.009 |
- |
4-Methylpyrazole |
apparent value |
681763 |
1.1.1.1 | 0.014 |
- |
5alpha-androstan-17beta-ol-3-one |
pH 7.3, 37°C, versus ethanol |
655206 |