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3.3 - 833
4-androstene-3,17-dione
20 - 417
5alpha-Androstan-17alpha-ol-3-one
0.03 - 4.5
5alpha-androstan-17beta-ol-3-one
1.5 - 122
5alpha-Androstan-3alpha-ol-17-one
0.05 - 0.65
5alpha-androstan-3beta,17beta-diol
83 - 8000
5beta-pregnane-20alpha-ol-3-one
60 - 8000
5beta-pregnane-3,20-dione
1 - 366
5beta-pregnane-3alpha,20alpha-diol
11.67 - 500
Epitestosterone
3.3
4-androstene-3,17-dione
mutant Y224D, pH 7.0, 25°C
105
4-androstene-3,17-dione
mutant Q222N, pH 7.0, 25°C
217
4-androstene-3,17-dione
mutant Y224F, pH 7.0, 25°C
833
4-androstene-3,17-dione
wild-type, pH 7.0, 25°C
20
5alpha-Androstan-17alpha-ol-3-one
mutant Q222N, pH 7.0, 25°C
160
5alpha-Androstan-17alpha-ol-3-one
mutant Y224F, pH 7.0, 25°C
417
5alpha-Androstan-17alpha-ol-3-one
wild-type, pH 7.0, 25°C
0.03
5alpha-androstan-17beta-ol-3-one
mutant Y224D, pH 7.0, 25°C
0.5
5alpha-androstan-17beta-ol-3-one
mutant Y224F, pH 7.0, 25°C
4.5
5alpha-androstan-17beta-ol-3-one
mutant Q222N, pH 7.0, 25°C
1.5
5alpha-Androstan-3alpha-ol-17-one
mutant Y224D, pH 7.0, 25°C
68.3
5alpha-Androstan-3alpha-ol-17-one
mutant Q222N, pH 7.0, 25°C
70
5alpha-Androstan-3alpha-ol-17-one
mutant Y224F, pH 7.0, 25°C
122
5alpha-Androstan-3alpha-ol-17-one
wild-type, pH 7.0, 25°C
0.05
5alpha-androstan-3beta,17beta-diol
mutant Y224D, pH 7.0, 25°C
0.167
5alpha-androstan-3beta,17beta-diol
mutant Y224F, pH 7.0, 25°C
0.65
5alpha-androstan-3beta,17beta-diol
mutant Q222N, pH 7.0, 25°C
83
5beta-pregnane-20alpha-ol-3-one
mutant Y224D, pH 7.0, 25°C
400
5beta-pregnane-20alpha-ol-3-one
mutant Q222N, pH 7.0, 25°C
2000
5beta-pregnane-20alpha-ol-3-one
wild-type, pH 7.0, 25°C
8000
5beta-pregnane-20alpha-ol-3-one
mutant Y224F, pH 7.0, 25°C
60
5beta-pregnane-3,20-dione
mutant Y224D, pH 7.0, 25°C
667
5beta-pregnane-3,20-dione
wild-type, pH 7.0, 25°C
1200
5beta-pregnane-3,20-dione
mutant Q222N, pH 7.0, 25°C
8000
5beta-pregnane-3,20-dione
mutant Y224F, pH 7.0, 25°C
1
5beta-pregnane-3alpha,20alpha-diol
mutant Y224D, pH 7.0, 25°C
65
5beta-pregnane-3alpha,20alpha-diol
mutant Q222N, pH 7.0, 25°C
125
5beta-pregnane-3alpha,20alpha-diol
mutant Y224F, pH 7.0, 25°C
366
5beta-pregnane-3alpha,20alpha-diol
wild-type, pH 7.0, 25°C
11.67
Epitestosterone
mutant Q222N, pH 7.0, 25°C
40
Epitestosterone
mutant Y224F, pH 7.0, 25°C
500
Epitestosterone
wild-type, pH 7.0, 25°C
1
lithocholic acid
mutant Y224D, pH 7.0, 25°C
183
lithocholic acid
mutant Q222N, pH 7.0, 25°C
400
lithocholic acid
mutant Y224F, pH 7.0, 25°C
467
lithocholic acid
wild-type, pH 7.0, 25°C