EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.22.B50 | 0.00015 |
- |
N-(3-fluorobenzyl)-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
731149 |
3.4.22.B50 | 0.0001712 |
- |
E-64 |
mutant enzyme S32T/A67Y, in 50 mM Na-acetate buffer pH 5.0, at 60°C |
732725 |
3.4.22.B50 | 0.0002137 |
- |
E-64 |
mutant enzyme S32T, in 50 mM Na-acetate buffer pH 5.0, at 60°C |
732725 |
3.4.22.B50 | 0.0002507 |
- |
E-64 |
mutant enzyme A67Y, in 50 mM Na-acetate buffer pH 5.0, at 60°C |
732725 |
3.4.22.B50 | 0.00032 |
- |
N-(1,3-benzodioxol-5-ylmethyl)-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
731149 |
3.4.22.B50 | 0.000349 |
- |
E-64 |
wild type enzyme, in 50 mM Na-acetate buffer pH 5.0, at 60°C |
732725 |
3.4.22.B50 | 0.00035 |
- |
N-[(2-methoxypyridin-4-yl)methyl]-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
731149 |
3.4.22.B50 | 0.00039 |
- |
N-[3-(acetylamino)benzyl]-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
731149 |
3.4.22.B50 | 0.00049 |
- |
N-(4-fluorobenzyl)-1-[(1R)-1-(naphthalen-1-yl)ethyl]piperidine-4-carboxamide |
pH and temperature not specified in the publication |
731149 |
3.4.22.B50 | 0.0006 |
- |
5-amino-2-methyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]benzamide |
pH and temperature not specified in the publication |
731149 |