EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.22.69 | 6e-18 |
- |
promazine |
in silico binding studies |
667918 |
| 3.4.22.69 | 8.7e-17 |
- |
lopinavir |
in silico binding studies |
667918 |
| 3.4.22.69 | 2.1e-16 |
- |
N-[3-[(E)-(tert-butoxyimino)methyl]-4-chlorophenyl]-2-methylfuran-3-carboxamide |
in silico binding studies |
667918 |
| 3.4.22.69 | 0.0000031 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-((S)-2-(2-(3-(dimethylamino)phenoxy)acetamido)-3-methylbutanamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.0000031 |
- |
N-[[3-(dimethylamino)phenoxy]acetyl]-L-valyl-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-L-leucinamide |
pH and temperature not specified in the publication |
731749 |
| 3.4.22.69 | 0.0000041 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-4-methyl-2-((S)-3-methyl-2-(2-phenoxyacetamido)butanamido)pentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.0000041 |
- |
N-[(benzyloxy)carbonyl]-L-valyl-N-[(2S)-1-(1,3-benzothiazol-2-yl)-1-oxo-3-[(3S)-2-oxopyrrolidin-3-yl]propan-2-yl]-L-leucinamide |
pH and temperature not specified in the publication |
731749 |
| 3.4.22.69 | 0.0000041 |
- |
Z-Val-Leu-Ala(-pyrrolidone-3-yl)-2-benzothiazole |
pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.0000063 |
- |
N-((S)-1-(((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)amino)-4-methyl-1-oxopentan-2-yl)-4-methoxy-1H-indole-2-carboxamide |
pH and temperature not specified in the publication |
731749 |
| 3.4.22.69 | 0.0000075 |
- |
1-[(1H-indol-5-ylcarbonyl)oxy]-1H-1,2,3-benzotriazole |
- |
679164 |
