EC Number   |
Authors |
Title |
Journal |
Organism |
|---|
   1.1.98.3 | Naik, M.; Humnabadkar, V.; Tantry, S.J.; Panda, M.; Narayan, A.; Guptha, S.; Panduga, V.; Manjrekar, P.; Jena, L.K.; Koushik, K.; Shanbhag, G.; Jatheendranath, S.; Manjunatha, M.R.; Gorai, G.; Bathula, C.; Rudrapatna, S.; Achar, V.; Sharma, S.; Ambady, A.; Hegde, N.; Mahadevaswamy, J.; Kaur, P.; Samb, S.a.m.b.a. |
4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity |
J. Med. Chem. |
Mycobacterium tuberculosis |
| 1.1.98.3 | Ribeiro, A.L.; Degiacomi, G.; Ewann, F.; Buroni, S.; Incandela, M.L.; Chiarelli, L.R.; Mori, G.; Kim, J.; Contreras-Dominguez, M.; Park, Y.S.; Han, S.J.; Brodin, P.; Valentini, G.; Rizzi, M.; Riccardi, G.; Pasca, M.R. |
Analogous mechanisms of resistance to benzothiazinones and dinitrobenzamides in Mycobacterium smegmatis |
PLoS ONE |
Mycolicibacterium smegmatis |
| 1.1.98.3 | Trefzer, C.; Skovierova, H.; Buroni, S.; Bobovska, A.; Nenci, S.; Molteni, E.; Pojer, F.; Pasca, M.; Makarov, V.; Cole, S.; Riccardi, G.; Mikusova, K.; Johnsson, K. |
Benzothiazinones are suicide inhibitors of mycobacterial decaprenylphosphoryl-beta-D-ribofuranose 2'-oxidase DprE1 |
J. Am. Chem. Soc. |
Mycolicibacterium smegmatis |
| 1.1.98.3 | Trefzer, C.; Rengifo-Gonzalez, M.; Hinner, M.J.; Schneider, P.; Makarov, V.; Cole, S.T.; Johnsson, K. |
Benzothiazinones: prodrugs that covalently modify the decaprenylphosphoryl-beta-D-ribose 2-epimerase DprE1 of Mycobacterium tuberculosis |
J. Am. Chem. Soc. |
Mycobacterium tuberculosis |
| 1.1.98.3 | Trefzer, C.; Rengifo-Gonzalez, M.; Hinner, M.J.; Schneider, P.; Makarov, V.; Cole, S.T.; Johnsson, K. |
Benzothiazinones: prodrugs that covalently modify the decaprenylphosphoryl-beta-D-ribose 2-epimerase DprE1 of Mycobacterium tuberculosis |
J. Am. Chem. Soc. |
Mycobacterium tuberculosis H37Rv |
| 1.1.98.3 | Foo, C.S.; Lechartier, B.; Kolly, G.S.; Boy-Roettger, S.; Neres, J.; Rybniker, J.; Lupien, A.; Sala, C.; Piton, J.; Cole, S.T. |
Characterization of DprE1-mediated benzothiazinone resistance in Mycobacterium tuberculosis |
Antimicrob. Agents Chemother. |
Mycobacterium tuberculosis |
| 1.1.98.3 | Foo, C.S.; Lechartier, B.; Kolly, G.S.; Boy-Roettger, S.; Neres, J.; Rybniker, J.; Lupien, A.; Sala, C.; Piton, J.; Cole, S.T. |
Characterization of DprE1-mediated benzothiazinone resistance in Mycobacterium tuberculosis |
Antimicrob. Agents Chemother. |
Mycobacterium tuberculosis H37Rv |
| 1.1.98.3 | Li, H.; Jogl, G. |
Crystal structure of decaprenylphosphoryl-beta-D-ribose 2'-epimerase from Mycobacterium smegmatis |
Proteins |
Mycolicibacterium smegmatis |
| 1.1.98.3 | Li, H.; Jogl, G. |
Crystal structure of decaprenylphosphoryl-beta-D-ribose 2'-epimerase from Mycobacterium smegmatis |
Proteins |
Mycolicibacterium smegmatis ATCC 700084 |
| 1.1.98.3 | Mikusova, K.; Huang, H.; Yagi, T.; Holsters, M.; Vereecke, D.; DHaeze, W.; Scherman, M.S.; Brennan, P.J.; McNeil, M.R.; Crick, D.C. |
Decaprenylphosphoryl arabinofuranose, the donor of the D-arabinofuranosyl residues of mycobacterial arabinan, is formed via a two-step epimerization of decaprenylphosphoryl ribose |
J. Bacteriol. |
Mycobacterium tuberculosis |
