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Literature summary for 3.4.22.1 extracted from

  • Mycek, M.J.
    Cathepsins (1970), Methods Enzymol., 19, 285-315.
No PubMed abstract available

Activating Compound

Activating Compound Comment Organism Structure
2,3-Dimercaptopropanol
-
Bos taurus
2-mercaptoethanol activates Rattus norvegicus
2-mercaptoethanol activates Bos taurus
2-mercaptoethylamine
-
Bos taurus
cysteine activates Rattus norvegicus
cysteine activates Bos taurus
glutathione activates Bos taurus
thiol compounds required for full activity Rattus norvegicus
thiol compounds required for full activity Bos taurus

Inhibitors

Inhibitors Comment Organism Structure
iodoacetamide
-
Bos taurus
N-ethylmaleimide no inhibition at 1 mM Bos taurus
p-chloromercuribenzoate
-
Bos taurus

Localization

Localization Comment Organism GeneOntology No. Textmining
lysosome
-
Bos taurus 5764
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
Proteins + H2O Rattus norvegicus
-
?
-
?
Proteins + H2O Bos taurus
-
?
-
?

Organism

Organism UniProt Comment Textmining
Bos taurus
-
-
-
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Bos taurus

Source Tissue

Source Tissue Comment Organism Textmining
spleen
-
Bos taurus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
benzoyl-arginine ethyl ester + H2O
-
Rattus norvegicus benzoyl-arginine + ethanol
-
?
benzoyl-arginine ethyl ester + H2O
-
Bos taurus benzoyl-arginine + ethanol
-
?
benzoyl-DL-argininamide + H2O
-
Rattus norvegicus benzoyl-DL-arginine + NH3
-
?
benzoyl-DL-argininamide + H2O
-
Bos taurus benzoyl-DL-arginine + NH3
-
?
Proteins + H2O
-
Rattus norvegicus ?
-
?
Proteins + H2O
-
Bos taurus ?
-
?