Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-mercaptoethanol | - |
Homo sapiens | |
benzyloxycarbonyl-Pro-prolinal | - |
Homo sapiens | |
Co2+ | - |
Homo sapiens | |
dithiothreitol | - |
Homo sapiens | |
EDTA | - |
Homo sapiens | |
Hg2+ | - |
Homo sapiens | |
additional information | resistant to: PMSF, thyorphan, E64 and phosphoramidon | Homo sapiens | |
o-phenanthroline | - |
Homo sapiens | |
p-hydroxymercuribenzoate | - |
Homo sapiens | |
PCMB | - |
Homo sapiens | |
Zn2+ | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00065 | - |
2-aminobenzoyl-FPQ-(N-(2,4-dinitrophenyl)ethylenediamine) | pH 8.0, 37°C | Homo sapiens | |
0.00074 | - |
2-aminobenzoyl-RPPGFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) | pH 8.0, 37°C | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
urine | - |
Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2-aminobenzoyl-FFQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | ? | - |
? | |
2-aminobenzoyl-FPQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | 2-aminobenzoyl-FP + Q-(N-(2,4-dinitrophenyl)ethylenediamine) | - |
? | |
2-aminobenzoyl-FSQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | ? | - |
? | |
2-aminobenzoyl-RPPGFQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | ? | - |
? | |
2-aminobenzoyl-RPPGFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | 2-aminobenzoyl-RPP + GFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) | - |
? | |
2-aminobenzoyl-SPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O | - |
Homo sapiens | ? | - |
? | |
Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg + H2O | as active as potentiator B | Homo sapiens | Lys-Arg-Pro-Pro + Gly-Phe-Ser-Pro-Phe-Arg | - |
? | |
Met-Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg + H2O | as active as potentiator B | Homo sapiens | Met-Lys-Arg-Pro-Pro + Gly-Phe-Ser-Pro-Phe-Arg | - |
? | |
additional information | no activity with Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2, pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr and pGly-His-Trp-Ser-tyr-Gly-leu-Arg-Pro-Gly-NH2 | Homo sapiens | ? | - |
? | |
pGlu-Gly-Leu-Pro-Pro-Arg-Pro + H2O | i.e. potentiator B | Homo sapiens | pGlu-Gly-Leu-Pro-Pro + Arg-Pro | - |
? | |
pGlu-Gly-Leu-Pro-Pro-Gly-Pro + H2O | i.e. potentiator C, as active as potentiator B | Homo sapiens | pGlu-Gly-Leu-Pro-Pro + Gly-Pro | - |
? | |
RPPGFSPFR + H2O | i.e. bradykinin, 90% of the activity with potentiator B, i.e. pGlu-Gly-Leu-Pro-Pro-Arg-Pro | Homo sapiens | ? | - |
? | |
RPPGFSPFR-amide + H2O | i.e. bradykinin, 70% of the activity with potentiator B, i.e. pGlu-Gly-Leu-Pro-Pro-Arg-Pro | Homo sapiens | RPP + GFSPFR-amide | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PE | - |
Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
6.5 | - |
reaction with 2-aminobenzoyl-FPQ-(N-(2,4-dinitrophenyl)ethylenediamine), and a second lower optimum at pH 8.0 | Homo sapiens |
8 | - |
reaction with bradykinin. And a second higher optimum at pH 6.5, reaction with 2-aminobenzoyl-FPQ-(N-(2,4-dinitrophenyl)ethylenediamine) | Homo sapiens |
9 | - |
reaction with 2-aminobenzoyl-RPPGFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) | Homo sapiens |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
7 | 9 | pH 7.0: about 55% of maximal activity, pH 9.0: about 30% of maximal activity, reaction with bradykinin | Homo sapiens |
8.5 | 10 | pH 8.5: about 40% of maximal activity, pH 10.0: about 80% of maximal activity, reaction with 2-aminobenzoyl-BKQRPPGFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) | Homo sapiens |