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Literature summary for 3.4.17.23 extracted from

  • Trask, A.J.; Groban, L.; Westwood, B.M.; Varagic, J.; Ganten, D.; Gallagher, P.E.; Chappell, M.C.; Ferrario, C.M.
    Inhibition of angiotensin-converting enzyme 2 exacerbates cardiac hypertrophy and fibrosis in Ren-2 hypertensive rats (2010), Am. J. Hypertens., 23, 687-693.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
MLN-4760
-
Rattus norvegicus

Metals/Ions

Metals/Ions Comment Organism Structure
Zn2+
-
Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
wild-type Ren-2 and transgenic hypertensive (mRen2)27 rats
-

Source Tissue

Source Tissue Comment Organism Textmining
cardiomyocyte
-
Rattus norvegicus
-
heart
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
7-methoxycoumarin-4-acetyl-Ala-Pro-Lys-(2,4-dinitrophenyl)-OH + H2O
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
ACE2
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
42
-
assay at Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7
-
assay at Rattus norvegicus

General Information

General Information Comment Organism
malfunction inhibition of angiotensin-converting enzyme 2 exacerbates cardiac hypertrophy and fibrosis in Ren-2 hypertensive rats Rattus norvegicus