EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.3.2.13 | -999 |
- |
more |
inhibition kinetic analysis |
759603 |
2.3.2.13 | -999 |
- |
more |
inhibition kinetics |
759606 |
2.3.2.13 | -999 |
- |
more |
inhibition kinetics, irreversible enzyme inactivation usually results in steady-state rates that are equal to zero independent of inhibitor concentration |
759049 |
2.3.2.13 | 0.00006 |
- |
Ac-P(6-diazo-5-oxo-L-norleucine)LPF-NH2 |
- |
689704 |
2.3.2.13 | 0.000075 |
- |
2-Iodoacetamide |
- |
689380 |
2.3.2.13 | 0.00014 |
- |
2-([3-(3-fluorophenyl)-5-(2-methoxyphenyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl]thio)acetohydrazide |
substrate N-methylcasein |
672218 |
2.3.2.13 | 0.00014 |
- |
2-[[3-(3-fluorophenyl)-5-(2-methoxyphenyl)-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl]thio]acetohydrazide |
transpeptidation of N,N-dimethylated casein by alphaN-Boc-Lys-NH-CH2-CH2-NH-dansyl |
672218 |
2.3.2.13 | 0.00016 |
- |
2-([3-(2-fluorophenyl)-4-oxo-5-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl]thio)acetohydrazide |
substrate N-methylcasein |
672218 |
2.3.2.13 | 0.00016 |
- |
2-[[3-(2-fluorophenyl)-4-oxo-5-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl]thio]acetohydrazide |
transpeptidation of N,N-dimethylated casein by alphaN-Boc-Lys-NH-CH2-CH2-NH-dansyl |
672218 |
2.3.2.13 | 0.00017 |
- |
2-[[3-(3-fluorophenyl)-4-oxo-5-phenyl-3,4,5,6,7,8-hexahydro[1]benzothieno[2,3-d]pyrimidin-2-yl]sulfanyl]acetohydrazide |
substrate N-methylcasein |
672218 |