Activating Compound | Comment | Organism | Structure |
---|---|---|---|
Calmodulin/Ca2+ | 0.01-0.2 mM, 3fold activation, inhibition above 0.3 mM, kinetics | Gallus gallus | |
Calmodulin/Ca2+ | 0.01-0.2 mM, 3fold activation, inhibition above 0.3 mM, kinetics | Homo sapiens | |
thrombin | slight activation | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
chlorpromazine | reverses calmodulin enzyme stimulation | Gallus gallus | |
chlorpromazine | reverses calmodulin enzyme stimulation | Homo sapiens | |
iodoacetamide | factor XIIIa; not inhibited in the absence of Ca2+, calmodulin regulated transglutaminases is not inhibited | Gallus gallus | |
iodoacetamide | factor XIIIa; not inhibited in the absence of Ca2+, calmodulin regulated transglutaminases is not inhibited | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.006 | - |
casein | plasma factor XII, actin | Gallus gallus | |
0.007 | - |
actin | platelet transglutaminase | Homo sapiens | |
0.011 | - |
casein | platelet transglutaminase | Homo sapiens | |
0.012 | - |
casein | gizzard transglutaminase | Gallus gallus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | requirement | Gallus gallus | |
Ca2+ | requirement | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
protein-bound gamma-glutamine + alkylamine | Gallus gallus | last enzyme in blood coagulation forming intermolecular gamma-glutamyl-epsilon-lysine crosslinks between fibrin molecules | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | Homo sapiens | last enzyme in blood coagulation forming intermolecular gamma-glutamyl-epsilon-lysine crosslinks between fibrin molecules | protein N5-alkylglutamine + NH3 | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Gallus gallus | - |
- |
- |
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
co-purified with alpha-actinin | Gallus gallus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
blood platelet | - |
Homo sapiens | - |
gizzard | smooth muscle | Gallus gallus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
monodansyl- cadaverine + actin | - |
Homo sapiens | ? | - |
? | |
N-(5-aminopentyl)-5-dimethylamino-1-naphthalenesulfonamide + casein | - |
Gallus gallus | ? | - |
? | |
N-(5-aminopentyl)-5-dimethylamino-1-naphthalenesulfonamide + casein | - |
Homo sapiens | ? | - |
? | |
N-(5-aminopentyl)-5-dimethylamino-1-naphthalenesulfonamide + F-actin | trivial name dansylcadaverine | Gallus gallus | ? | - |
? | |
N-(5-aminopentyl)-5-dimethylamino-1-naphthalenesulfonamide + F-actin | trivial name dansylcadaverine | Homo sapiens | ? | - |
? | |
protein-bound gamma-glutamine + alkylamine | donors: gamma-carboxamide groups of protein-bound glutamine, acceptors: epsilon-amino groups of protein-bound lysine | Gallus gallus | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | donors: gamma-carboxamide groups of protein-bound glutamine, acceptors: epsilon-amino groups of protein-bound lysine | Homo sapiens | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | forms intramolecular isopeptide bonds between fibrin molecules | Gallus gallus | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | forms intramolecular isopeptide bonds between fibrin molecules | Homo sapiens | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | last enzyme in blood coagulation forming intermolecular gamma-glutamyl-epsilon-lysine crosslinks between fibrin molecules | Gallus gallus | protein N5-alkylglutamine + NH3 | - |
? | |
protein-bound gamma-glutamine + alkylamine | last enzyme in blood coagulation forming intermolecular gamma-glutamyl-epsilon-lysine crosslinks between fibrin molecules | Homo sapiens | protein N5-alkylglutamine + NH3 | - |
? |