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BRENDA support

Literature summary for 1.1.1.B40 extracted from

  • Gong, R.; Morris, D.J.; Brem, A.S.
    Human renal 11beta-hydroxysteroid dehydrogenase 1 functions and co-localizes with COX-2 (2008), Life Sci., 82, 631-637.
    View publication on PubMed

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.0000102
-
NAD+ kidney homogenate, pH and temperature not specified in the publication Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
kidney similar amounts of protein for both isoform 11beta-HSD1 and 11beta-HSD2. 11beta-HSD1 functions as a dehydrogenase with no significant reverse reductase activity and colocalizes with cyclooxygenase COX-2 in proximal tubule cells. No colocalization of COX-2 with isoform 11beta-HSD2 in cortical collecting duct Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
cortisol + NAD+
-
Homo sapiens cortisone + NADH
-
?

Synonyms

Synonyms Comment Organism
11beta-HSD2
-
Homo sapiens
11beta-hydroxysteroid dehydrogenase 2
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
NAD+
-
Homo sapiens