Inhibitors | Comment | Organism | Structure |
---|---|---|---|
glycyrrhetinic acid | strong inhibition of isozyme 11beta-HSD2 | Rhinella arenarum |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00013 | - |
corticosterone | pH 8.0, 28°C, isozyme 11beta-HSD2, R period | Rhinella arenarum | |
0.00014 | - |
corticosterone | pH 8.0, 28°C, isozyme 11beta-HSD2, PR period | Rhinella arenarum | |
0.00028 | - |
corticosterone | pH 8.0, 28°C, isozyme 11beta-HSD2, P period | Rhinella arenarum |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | isozyme 11beta-HSD2 | Rhinella arenarum | - |
- |
mitochondrion | isozyme 11beta-HSD2 | Rhinella arenarum | 5739 | - |
additional information | subcellular localization of isozyme 11beta-HSD2, overview, isozyme 11beta-HSD2 activity and plasma corticosterone are determined in toads from pre- (PR), post- (P), and reproductive (R) periods, overview | Rhinella arenarum | - |
- |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
corticosterone + NAD+ | Rhinella arenarum | isozyme 11beta-HSD2 | 11-dehydrocorticosterone + NADH + H+ | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rhinella arenarum | - |
isozyme 11beta-HSD2 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
additional information | isozyme 11beta-HSD2activity and plasma corticosterone are determined in toads from pre- (PR), post- (P), and reproductive (R) periods, activity is highest in P period, overview | Rhinella arenarum | - |
testis | isozyme 11beta-HSD2 | Rhinella arenarum | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
isozyme 11beta-HSD2 activity and plasma corticosterone are determined in toads from pre- (PR), post- (P), and reproductive (R) periods, activity is highest in P period, overview | Rhinella arenarum |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
corticosterone + NAD+ | isozyme 11beta-HSD2 | Rhinella arenarum | 11-dehydrocorticosterone + NADH + H+ | - |
? |
Synonyms | Comment | Organism |
---|---|---|
11 beta-hydroxysteroid dehydrogenase | - |
Rhinella arenarum |
11beta-HSD2 | - |
Rhinella arenarum |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
28 | - |
assay at | Rhinella arenarum |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
8 | - |
assay at | Rhinella arenarum |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
NAD+ | isozyme 11beta-HSD2, dependent on | Rhinella arenarum |