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0.000064
(+/-)-2-((cyclohexylmethyl)amino)-5-ethyl-5-methyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000034
(+/-)-2-((cyclohexylmethyl)amino)-5-methyl-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000024
(+/-)-2-(1-adamantylamino)-5-ethyl-5-methyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000024
(+/-)-2-(1-adamantylamino)-5-methyl-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000082
(+/-)-2-(cycloheptylamino)-5-ethyl-5-methyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000032
(+/-)-2-(cycloheptylamino)-5-methyl-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000126
(+/-)-2-(cyclohexylamino)-5-ethyl-5-methyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000055
(+/-)-2-(cyclohexylamino)-5-methyl-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000047
(+/-)-2-(cyclooctylamino)-5-ethyl-5-methyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000028
(+/-)-2-(cyclooctylamino)-5-methyl-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000073
(+/-)-5-ethyl-5-methyl-2-(1-norbornylamino)-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000013
(+/-)-5-ethyl-5-methyl-2-(3-noradamantylamino)-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000372
(+/-)-5-ethyl-5-methyl-2-(7-norbornylamino)-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000058
(+/-)-5-ethyl-5-methyl-2-[(2,2,3,3-tetramethylcyclopropyl)amino]-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000025
(+/-)-5-methyl-2-(1-norbornylamino)-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000012
(+/-)-5-methyl-2-(3-noradamantylamino)-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000149
(+/-)-5-methyl-2-(7-norbornylamino)-5-propyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000038
(+/-)-5-methyl-5-propyl-2-[(2,2,3,3-tetramethylcyclopropyl)amino]-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.01874 - 0.02268
(-)-epigallocatechin 3-gallate
0.0000472
(R)-2-((1R,2R,4S)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.00077
(R)-2-((1R,2R,4S)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.0000306
(R)-2-((1S,2S,4R)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000329
(R)-2-((1S,2S,4R)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.0000278
(S)-2-((1R,2R,4S)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000227
(S)-2-((1R,2R,4S)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.0000128
(S)-2-((1S,2S,4R)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000012
(S)-2-((1S,2S,4R)-bicyclo[2.2.1]heptan-2-ylamino)-5-isopropylthiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000028
2-(1-adamantylamino)-1-thia-3-azaspiro[4.4]non-2-en-4-one
pH and temperature not specified in the publication
0.00002
2-(1-adamantylamino)-5,5-diethyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.000003
2-(3-noradamantylamino)-1-thia-3-azaspiro[4.4]non-2-en-4-one
pH and temperature not specified in the publication
0.000287
2-(6-[[(3-chloro-2-methylphenyl)sulfonyl]amino]pyridin-2-yl)-N,N-diethylacetamide
-
pH not specified in the publication, temperature not specified in the publication
0.000058
2-(bicyclo[2.2.1]hept-2-ylamino)-5-(propan-2-yl)-1,3-thiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000014
2-(cyclooctylamino)-1-thia-3-azaspiro[4.4]non-2-en-4-one
pH and temperature not specified in the publication
0.000026
2-(cyclooctylamino)-5,5-diethyl-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.0000173
2-[(1S,2S,4R)-bicyclo[2.2.1]hept-2-ylamino]-5-methyl-5-(propan-2-yl)-1,3-thiazol-4(5H)-one
pH not specified in the publication, temperature not specified in the publication
0.000169
3-chloro-2-methyl-N-(6-methylpyridin-2-yl)benzenesulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000169
3-chloro-2-methyl-N-[6-[2-oxo-2-(piperidin-1-yl)ethyl]pyridin-2-yl]benzenesulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000058
4'-chloro-N-(6-methylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000019
4'-cyano-N-(6-cyclopropylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000066
4'-cyano-N-(6-ethylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000004
4'-cyano-N-(6-methylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000048
4'-cyano-N-[6-(ethylamino)pyridin-2-yl]biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000098
4'-cyano-N-[6-(methylamino)pyridin-2-yl]biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0000017
4'-cyano-N-[6-(propan-2-yl)pyridin-2-yl]biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.00002
4'-fluoro-N-(6-methylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000062
4'-methyl-N-(6-methylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000013
5,5-diethyl-2-(3-noradamantylamino)-1,3-thiazol-4-(5H)-one
pH and temperature not specified in the publication
0.00005 - 0.003
arylsulfoamidothiazole
0.0016
fenofibrate
-
82% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.0091
fenofibric acid cyclohexyl ester
-
54% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.0034
fenofibric acid ethylester
-
85% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.0031
fenofibric acid isobutylester
-
75% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.009
fenofibric acid isopropyl amide
-
54% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.0041
fenofibric acid n-butylester
-
64% inhibition at 0.01 mM, cell-based assay, pH not specified in the publication, temperature not specified in the publication
0.0000049 - 0.000014
glycyrrhetinic acid
0.000108
N-(6-methylpyridin-2-yl)-4-(trifluoromethyl)benzenesulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000048
N-(6-methylpyridin-2-yl)biphenyl-4-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.000084
N-(6-methylpyridin-2-yl)naphthalene-2-sulfonamide
-
pH not specified in the publication, temperature not specified in the publication
0.0396
resveratrol
-
at pH 7.4 and 37°C
additional information
N-(6-aminopyridin-2-yl)-4'-cyanobiphenyl-4-sulfonamide
-
Ki below 0.000001 mM, pH not specified in the publication, temperature not specified in the publication
0.01874
(-)-epigallocatechin 3-gallate
purified enzyme, at pH 7.4 and 37°C
0.02268
(-)-epigallocatechin 3-gallate
unpurified enzyme, at pH 7.4 and 37°C
0.00005
arylsulfoamidothiazole
-
0.003
arylsulfoamidothiazole
-
above
0.003
arylsulfoamidothiazole
-
above
0.0000049
glycyrrhetinic acid
-
37°C, pH 9.0, inhibition of cortisol oxidation
0.000005
glycyrrhetinic acid
-
vs. cortisol
0.00001
glycyrrhetinic acid
-
vs. 4-methylnitrosamine-1-(3-pyridiyl)-1-butanone
0.000014
glycyrrhetinic acid
-
37°C, pH 9.0, inhibition of cortisone reduction
0.000014
glycyrrhetinic acid
-
vs. cortisone